Fundraising Fox

Dario Doller

Founder

Co-founder at Modulate Bio

New York City Metropolitan Area

FoundedModulate Bio

About

Dario Doller is Chief Scientific Officer at Modulate Bio, with expertise in allosteric drug discovery targeting GPCRs, ion channels, and enzymes for CNS, metabolic, and cardiovascular indications. Over a 30-year career in pharma and biotech, he contributed to the FDA-approved drug Vorapaxar and to four additional clinical-stage compounds (CTP-692, NGD-4715, and Lu AF09535), and edited two books, Allosterism in Drug Discovery (RSC, 2017) and Trends in CNS Drug Discovery (Wiley, 2025). His background spans medicinal chemistry, CNS chemical biology, pharmacokinetics, and in vitro and in vivo pharmacology.

Co-founder at Modulate Bio

Intro paths

In turn, Dario can intro founders to Modulate Bio's investors below.

Modulate Bio's investors · 1

Co-founders at Modulate Bio

KHKevin Hodgetts
Kevin HodgettsFounding Lab / Co-founder

Experience

  1. Modulate BioChief Scientific Officer (CSO)current2023 — presentMassachusetts, United States
  2. Nabu TherapeuticsVP of Medicinal Chemistrycurrent2025 — presentSan Francisco Bay Area
  3. Babylon BiosciencesDiscovery Teamcurrent2025 — presentSan Francisco Bay Area
  4. Alcyoneus ScienceWorksEarly discovery consulting2015 — 2025NJ, USA
  5. iNeuro Therapeutics IncVP Chemistry2022 — 2023Cambridge, Massachusetts, United States
  6. Lucy TherapeuticsVP, Drug Discovery2021 — 2022Cambridge, Massachusetts, United States
  7. Sunovion PharmaceuticalsDirector, Medicinal Chemistry2019 — 2021Marlborough, MA
  8. Sage TherapeuticsSenior Director, Head of Exploratory Research2017 — 2019Cambridge, MA
  9. CoNCERT Pharmaceuticals, Inc.Senior Director, Deuterium Platform2016 — 2017Greater Boston
  10. LundbeckChemical Biology, Global Head2014 — 2015Paramus, NJ
  11. LundbeckDirector, Global Project Leader (Discovery Chemistry & DMPK Department)2011 — 2014Paramus, NJ
  12. LundbeckDirector, Medicinal Chemistry (Chemical and Pharmacokinetic Sciences Department)2010 — 2011
  13. LundbeckDirector, Medicinal Chemistry2006 — 2010
  14. Neurogen CorporationAssociate Director2000 — 2006
  15. GliatechSenior Scientist1999 — 2000
  16. 3-Dimensional PharmaceuticalsGroup Leader1998 — 1999
  17. Schering-Plough Research InstituteSenior Scientist1994 — 1998
  18. Rohm and HaasResearch Scientist1992 — 1994Springhouse, PA
  19. Texas A&M UniversityPost-doc1989 — 1992

Skills & more

Biomarker Discovery6Translational MedicineBusiness DevelopmentAnalytical SkillsGritStructural BiologyScenario PlanningOut-licensingIn-licensingDevelopment ProgramsDrug Discovery99Medicinal Chemistry99
+12 moreDrug DesignPharmacologyDrug DevelopmentBiotechnologyChemistryNeuroscienceDMPKPharmacokineticsGPCRsAssay DevelopmentCollaborative Problem SolvingCreative Solutions

Languages Spanish

From Dario's professional profile.

Frequently asked questions

Who is Dario Doller?
Dario Doller is Chief Scientific Officer at Modulate Bio, with expertise in allosteric drug discovery targeting GPCRs, ion channels, and enzymes for CNS, metabolic, and cardiovascular indications. Over a 30-year career in pharma and biotech, he contributed to the FDA-approved drug Vorapaxar and to four additional clinical-stage compounds (CTP-692, NGD-4715, and Lu AF09535), and edited two books, Allosterism in Drug Discovery (RSC, 2017) and Trends in CNS Drug Discovery (Wiley, 2025). His background spans medicinal chemistry, CNS chemical biology, pharmacokinetics, and in vitro and in vivo pharmacology.
Where does Dario Doller work?
Dario Doller is Co-founder of Modulate Bio.
What companies did Dario Doller found?
Dario Doller founded Modulate Bio.
Where did Dario Doller go to school?
Dario Doller studied at University of Buenos Aires (Doctor of Philosophy - PhD, Chemical Sciences); University of Buenos Aires (Licentiate degree, Organic Chemistry).

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